Inhibitor Scaffolds for 2-Oxoglutarate-Dependent Histone Lysine Demethylases-Reference-Cited by-同舟云学术

Inhibitor Scaffolds for 2-Oxoglutarate-Dependent Histone Lysine Demethylases

Published:2008-10-23 Issue:22 Volume:51 Page:7053-7056
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Rose Nathan R.¹,Ng Stanley S.¹,Mecinović Jasmin¹,Liénard Benoît M.R.¹,Bello Simon H.¹,Sun Zhe¹,McDonough Michael A.¹,Oppermann Udo¹,Schofield Christopher J.¹

Affiliation:

1. The Department of Chemistry and the Oxford Centre for Integrative Systems Biology, Chemistry Research Laboratory, University of Oxford, 12 Mansfield Road, Oxford, OX1 3TA, United Kingdom, Structural Genomics Consortium, University of Oxford, Old Road Campus Roosevelt Drive, Headington, OX3 7DQ, United Kingdom, The Botnar Research Centre, Oxford Biomedical Research Unit, Oxford, OX3 7LD, United Kingdom

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm800936s

Reference16 articles.

1. Regulation of histone methylation by demethylimination and demethylation

2. Dimethyl sulfoxide to vorinostat: development of this histone deacetylase inhibitor as an anticancer drug

3. Histone H3 Lysine 4 Demethylation Is a Target of Nonselective Antidepressive Medications

4. Specificity and mechanism of JMJD2A, a trimethyllysine-specific histone demethylase

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