γ-Amino-Substituted Analogues of 1-[(S)-2,4-Diaminobutanoyl]piperidine as Highly Potent and Selective Dipeptidyl Peptidase II Inhibitors-Reference-Cited by-同舟云学术

γ-Amino-Substituted Analogues of 1-[(S)-2,4-Diaminobutanoyl]piperidine as Highly Potent and Selective Dipeptidyl Peptidase II Inhibitors

Published:2004-04-07 Issue:11 Volume:47 Page:2906-2916
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Senten Kristel¹,Van der Veken Pieter¹,De Meester Ingrid¹,Lambeir Anne-Marie¹,Scharpé Simon¹,Haemers Achiel¹,Augustyns Koen¹

Affiliation:

1. Department of Medicinal Chemistry and Department of Medical Biochemistry, University of Antwerp, Universiteitsplein 1, B-2610 Antwerp, Belgium

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm031122f

Reference32 articles.

1. Barrett, A. J., Rawlings, N. D., Woessner, J. F., Eds. Introduction: Clan SC Containing Peptidases with the α/β Hydrolase Fold.Handbook ofProteolytic Enzymes; Academic Press: San Diego, CA, 1998; Section 124, pp 369−372.

2. Prolyl peptidases: a serine protease subfamily with high potential for drug discovery

3. Dipeptidyl peptidase IV-like molecules: homologous proteins or homologous activities?

4. Villhauer, E. B.; Coppola, G. M.; Hughes, T. E. DPP−IV Inhibition and Therapeutic Potential.Annual Reports in Medicinal Chemistry; Academic Press: San Diego, CA, 2001; Vol. 36, pp 191−200.

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