Engineering Galanin Analogues That Discriminate between GalR1 and GalR2 Receptor Subtypes and Exhibit Anticonvulsant Activity following Systemic Delivery-Reference-Cited by-同舟云学术

Engineering Galanin Analogues That Discriminate between GalR1 and GalR2 Receptor Subtypes and Exhibit Anticonvulsant Activity following Systemic Delivery

Published:2010-02-01 Issue:4 Volume:53 Page:1871-1875
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Robertson Charles R.¹,Scholl Erika Adkins²,Pruess Timothy H.²,Green Brad R.¹,White H. Steve²,Bulaj Grzegorz¹

Affiliation:

1. Department of Medicinal Chemistry

2. Department of Pharmacology and Toxicology

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm9018349

Reference19 articles.

1. Regulation of Kindling Epileptogenesis by Hippocampal Galanin Type 1 and Type 2 Receptors: The Effects of Subtype-Selective Agonists and the Role of G-Protein-Mediated Signaling

2. Galanin – 25 years with a multitalented neuropeptide

3. Galanin – 25 years with a multitalented neuropeptide

4. Galmic, a nonpeptide galanin receptor agonist, affects behaviors in seizure, pain, and forced-swim tests

5. Design, Synthesis, and Characterization of High-Affinity, Systemically-Active Galanin Analogues with Potent Anticonvulsant Activities

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