Synthesis and Evaluation of Bivalent NDP-α-MSH(7) Peptide Ligands for Binding to the Human Melanocortin Receptor 4 (hMC4R)-Reference-Cited by-同舟云学术

Synthesis and Evaluation of Bivalent NDP-α-MSH(7) Peptide Ligands for Binding to the Human Melanocortin Receptor 4 (hMC4R)

Published:2007-06-26 Issue:4 Volume:18 Page:1101-1109
ISSN:1043-1802
Container-title:Bioconjugate Chemistry
language:en
Short-container-title:Bioconjugate Chem.

Author:

Handl Heather L.¹,Sankaranarayanan Rajesh¹,Josan Jatinder S.¹,Vagner Josef¹,Mash Eugene A.¹,Gillies Robert J.¹,Hruby Victor J.¹

Affiliation:

1. Department of Chemistry, University of Arizona, Tucson, Arizona 85721, and Departments of Radiology, Biochemistry, and Molecular Biophysics, Arizona Cancer Center, Tucson, Arizona 85724

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Pharmaceutical Science,Pharmacology,Biomedical Engineering,Bioengineering,Biotechnology

Link

https://pubs.acs.org/doi/pdf/10.1021/bc0603642

Reference27 articles.

1. Peptide Receptors as Molecular Targets for Cancer Diagnosis and Therapy

2. Novel targeting strategy based on multimeric ligands for drug delivery and molecular imaging: homooligomers of α-MSH

3. Biebermann, H., Krude, H., Elsner, A., Chubanov, V., Gudermann, T., and Gruters, A. (2003) Autosomal-dominant mode of inheritance of a melanocortin-4 receptor mutation in a patient with severe early-onset obesity is due to a dominant-negative effect caused by receptor dimerization.Diabetes 52, 2984−2988.

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