A Potent, Selective, and Cell-Active Inhibitor of Human Type I Protein Arginine Methyltransferases

Author:

Eram Mohammad S.1,Shen Yudao2,Szewczyk Magdalena M.1,Wu Hong1,Senisterra Guillermo1,Li Fengling1,Butler Kyle V.2,Kaniskan H. Ümit2,Speed Brandon A.2,dela Seña Carlo1,Dong Aiping1,Zeng Hong1,Schapira Matthieu13,Brown Peter J.1,Arrowsmith Cheryl H.14,Barsyte-Lovejoy Dalia1,Liu Jing2,Vedadi Masoud13,Jin Jian2

Affiliation:

1. Structural Genomics Consortium, University of Toronto, Toronto, Ontario M5G 1L7, Canada

2. Departments of Structural and Chemical Biology, Oncological Sciences, and Pharmacology and Systems Therapeutics, Icahn School of Medicine at Mount Sinai, New York, New York 10029, United States

3. Department of Pharmacology and Toxicology, University of Toronto, Toronto, Ontario M5S 1A8, Canada

4. Princess Margaret Cancer Centre and Department of Medical Biophysics, University of Toronto, Toronto, Ontario M5G 2M9, Canada

Funder

European Commission

Wellcome Trust

American Cancer Society

National Institute of General Medical Sciences

Structural Genomics Consortium

European Federation of Pharmaceutical Industries and Associations

Publisher

American Chemical Society (ACS)

Subject

Molecular Medicine,General Medicine,Biochemistry

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