Discovery and SAR of Natural-Product-Inspired RXR Agonists with Heterodimer Selectivity to PPARδ-RXR-Reference-Cited by-同舟云学术

Discovery and SAR of Natural-Product-Inspired RXR Agonists with Heterodimer Selectivity to PPARδ-RXR

Published:2020-05-06 Issue:6 Volume:15 Page:1526-1534
ISSN:1554-8929
Container-title:ACS Chemical Biology
language:en
Short-container-title:ACS Chem. Biol.

Author:

Nakashima Ken-ichi¹^ORCID,Yamaguchi Eiji^ORCID,Noritake Chihaya¹,Mitsugi Yukari,Goto Mayuki,Hirai Takao¹,Abe Naohito,Sakai Eiji,Oyama Masayoshi,Itoh Akichika^ORCID,Inoue Makoto¹

Affiliation:

1. Laboratory of Medicinal Resources, School of Pharmacy, Aichi Gakuin University, 1-100 Kusumoto-cho, Chikusa-ku, Nagoya 464-8650, Japan

Funder

Japan Society for the Promotion of Science

Publisher

American Chemical Society (ACS)

Subject

Molecular Medicine,General Medicine,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acschembio.0c00146

Reference40 articles.

1. A Unified Nomenclature System for the Nuclear Receptor Superfamily

2. Overview of Nomenclature of Nuclear Receptors

3. A revisited version of the apo structure of the ligand-binding domain of the human nuclear receptor retinoic X receptor α

4. A canonical structure for the ligand-binding domain of nuclear receptors

5. Crystal structure of the RAR-γ ligand-binding domain bound to all-trans retinoic acid

Cited by 7 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Osteoprotegerin mediates adipogenesis in obesity;Journal of Advanced Research;2024-08

2. Mechanisms of obesogens and their impact on adipose tissue, hormones, and inflammation;Journal of Medical Science;2024-03-18

3. Mesoporous Tio2 Supported Synthesis of Aryl Propionic Acid Derivatives, and Mild Peroxides, Organometallic Catalyst Free Oxidative Cleavage of C=C in Electron Deficient Olefins;2024

4. Regulation of adipogenesis through retinoid X receptor and/or peroxisome proliferator-activated receptor by designed lignans based on natural products in 3T3–L1 cells;Journal of Natural Medicines;2023-01-06

5. Use of GAL4 factor-based yeast assay to quantify the effects of xenobiotics on RXR homodimer and RXR/PPAR heterodimer in scallop Chlamys farreri;Science of The Total Environment;2022-12