Kinetic and Thermodynamic Insights into Agonist Interactions with the Parathyroid Hormone Receptor-1 from a New NanoBRET Assay
Author:
Affiliation:
1. Department of Chemistry, University of Wisconsin - Madison, Madison, Wisconsin53706United States
2. Endocrine Unit, Massachusetts General Hospital and Harvard Medical School, Boston, Massachusetts02114United States
Funder
National Institutes of Health
University of Wisconsin-Madison
National Science Foundation
Publisher
American Chemical Society (ACS)
Subject
Molecular Medicine,General Medicine,Biochemistry
Link
https://pubs.acs.org/doi/pdf/10.1021/acschembio.2c00595
Reference42 articles.
1. International Union of Basic and Clinical Pharmacology. XCIII. The Parathyroid Hormone Receptors—Family B G Protein–Coupled Receptors
2. PTH receptor-1 signalling—mechanistic insights and therapeutic prospects
3. PTH/PTHrP Receptor Signaling, Allostery, and Structures
4. Teriparatide
5. Abaloparatide: First Global Approval
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