A Chemical Biological Approach to Study G Protein-Coupled Receptors: Labeling the Adenosine A<sub>1</sub> Receptor Using an Electrophilic Covalent Probe-Reference-Cited by-同舟云学术

A Chemical Biological Approach to Study G Protein-Coupled Receptors: Labeling the Adenosine A₁ Receptor Using an Electrophilic Covalent Probe

Published:2022-10-24 Issue:11 Volume:17 Page:3131-3139
ISSN:1554-8929
Container-title:ACS Chemical Biology
language:en
Short-container-title:ACS Chem. Biol.

Author:

Beerkens Bert L. H.¹,Koç Çağla¹,Liu Rongfang¹,Florea Bogdan I.²^ORCID,Le Dévédec Sylvia E.¹^ORCID,Heitman Laura H.¹³,IJzerman Adriaan P.¹^ORCID,van der Es Daan¹^ORCID

Affiliation:

1. Division of Drug Discovery and Safety, Leiden Academic Centre for Drug Research, Leiden University, Einsteinweg 55, 2333 CC Leiden, The Netherlands

2. Department of Bioorganic Synthesis, Leiden Institute of Chemistry, Leiden University, Einsteinweg 55, 2333 CC Leiden, The Netherlands

3. Oncode Institute, 2333 CC Leiden, The Netherlands

Publisher

American Chemical Society (ACS)

Subject

Molecular Medicine,General Medicine,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acschembio.2c00589

Reference53 articles.

1. International Union of Basic and Clinical Pharmacology. LXXXI. Nomenclature and Classification of Adenosine Receptors—An Update

2. International Union of Basic and Clinical Pharmacology. CXII: Adenosine Receptors: A Further Update

3. The adenosine pathway in immuno-oncology