Residue-Based Preorganization of BH3-Derived α/β-Peptides: Modulating Affinity, Selectivity and Proteolytic Susceptibility in α-Helix Mimics-Reference-Cited by-同舟云学术

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Residue-Based Preorganization of BH3-Derived α/β-Peptides: Modulating Affinity, Selectivity and Proteolytic Susceptibility in α-Helix Mimics

Published:2015-05-07 Issue:7 Volume:10 Page:1667-1675
ISSN:1554-8929
Container-title:ACS Chemical Biology
language:en
Short-container-title:ACS Chem. Biol.

Author:

Peterson-Kaufman Kimberly J.¹,Haase Holly S.¹,Boersma Melissa D.¹,Lee Erinna F.²³,Fairlie W. Douglas²³,Gellman Samuel H.¹

Affiliation:

1. Department of Chemistry, University of Wisconsin, 1101 University Ave., Madison, Wisconsin 53706, United States

2. Structural Biology Division, The Walter and Eliza Hall Institute for Medical Research, 1G Royal Parade, Parkville, Victoria 3052, Australia

3. Department of Medical Biology, The University of Melbourne, Parkville, Victoria 3010, Australia

Funder

National Health and Medical Research Council

National Institute of General Medical Sciences

Publisher

American Chemical Society (ACS)

Subject

Molecular Medicine,General Medicine,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acschembio.5b00109

Reference57 articles.

1. Assessment of helical interfaces in protein–protein interactions

2. Systematic Analysis of Helical Protein Interfaces Reveals Targets for Synthetic Inhibitors

3. Assessing Helical Protein Interfaces for Inhibitor Design

4. Inhibition of α-helix-mediated protein–protein interactions using designed molecules

5. Terphenyl‐Based Helical Mimetics That Disrupt the p53/HDM2 Interaction

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