Selective and Potent PROTAC Degraders of c-Src Kinase-Reference-Cited by-同舟云学术

Selective and Potent PROTAC Degraders of c-Src Kinase

Published:2023-12-19 Issue:1 Volume:19 Page:110-116
ISSN:1554-8929
Container-title:ACS Chemical Biology
language:en
Short-container-title:ACS Chem. Biol.

Author:

Mao Wuxiang¹,Vandecan Nathalie M.¹,Bingham Christopher R.¹,Tsang Pui Ki¹,Ulintz Peter²,Sexton Rachel¹,Bochar Daniel A.¹,Merajver Sofia D.²,Soellner Matthew B.¹²^ORCID

Affiliation:

1. Department of Chemistry, University of Michigan, 930 N. University Avenue, Ann Arbor, Michigan 48109, United States

2. Department of Internal Medicine, University of Michigan, 1500 E. Medical Avenue, Ann Arbor, Michigan 48109, United States

Funder

National Institute of General Medical Sciences

Publisher

American Chemical Society (ACS)

Subject

Molecular Medicine,General Medicine,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acschembio.3c00548

Reference33 articles.

1. A historical overview of protein kinases and their targeted small molecule inhibitors

2. The ErbB/HER family of protein-tyrosine kinases and cancer

3. Src protein-tyrosine kinase structure, mechanism, and small molecule inhibitors

4. Structural Basis for the Non-catalytic Functions of Protein Kinases

5. The secret life of kinases: insights into non-catalytic signalling functions from pseudokinases

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