Development of a Benzothiazole Scaffold-Based Androgen Receptor N-Terminal Inhibitor for Treating Androgen-Responsive Prostate Cancer

Author:

Kuznik Nane C.1,Solozobova Valeria1,Jung Nicole2ORCID,Gräßle Simone2,Lei Qing1,Lewandowski Eric M.3,Munuganti Ravi4,Zoubeidi Amina45,Chen Yu3,Bräse Stefan26,Cato Andrew C. B.1ORCID

Affiliation:

1. Institute of Biological and Chemical Systems, Biological Information Processing, Karlsruhe Institute of Technology, 76344 Eggenstein-Leopoldshafen, Germany

2. Institute of Biological and Chemical Systems, Functional Molecular Systems, Karlsruhe Institute of Technology, 76344 Eggenstein-Leopoldshafen, Germany

3. Department of Molecular Medicine, Morsani College of Medicine, University of South Florida, Tampa, Florida 33612-4799, United States

4. Vancouver Prostate Centre, Vancouver, BC V6H 3Z6, Canada

5. Department of Urology, Faculty of Medicine, University of British Columbia, Vancouver, BC V5Z 1M9, Canada

6. Institute of Organic Chemistry, Karlsruhe Institute of Technology, 76131 Karlsruhe, Germany

Funder

Deutsche Forschungsgemeinschaft

Wilhelm Sander-Stiftung

Prostate Cancer Foundation

Publisher

American Chemical Society (ACS)

Subject

Molecular Medicine,General Medicine,Biochemistry

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