Design and Synthesis of Novel Indole β-Diketo Acid Derivatives as HIV-1 Integrase Inhibitors-Reference-Cited by-同舟云学术

Design and Synthesis of Novel Indole β-Diketo Acid Derivatives as HIV-1 Integrase Inhibitors

Published:2004-09-16 Issue:21 Volume:47 Page:5298-5310
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Sechi Mario¹,Derudas Massimiliano¹,Dallocchio Roberto¹,Dessì Alessandro¹,Bacchi Alessia¹,Sannia Luciano¹,Carta Fabrizio¹,Palomba Michele¹,Ragab Omar¹,Chan Carney¹,Shoemaker Robert¹,Sei Shizuko¹,Dayam Raveendra¹,Neamati Nouri¹

Affiliation:

1. Dipartimento Farmaco Chimico Tossicologico, Università di Sassari, Via Muroni 23/A, 07100 Sassari, Italy, CNR-Istituto di Chimica Biomolecolare, sez. di Sassari, Trav. La Crucca 3, reg. Baldinca, 07040 Li Punti, Italy, Dipartimento di Chimica Generale ed Inorganica, Chimica Analitica, Chimica Fisica, Università di Parma, Parco Area delle Scienze 17/A, 43100 Parma, Italy, Department of Pharmaceutical Sciences, School of Pharmacy, University of Southern California, 1985 Zonal Avenue, PSC 304, Los Angeles,...

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm049944f

Reference62 articles.

1. Strategies in the design of antiviral drugs

2. HIV chemotherapy

3. Activities of human immunodeficiency virus (HIV) integration protein in vitro: specific cleavage and integration of HIV DNA.

4. Brown, P. O.Integration; Cold Spring Harbor Press: Cold Spring Harbor, 1999.

Cited by 135 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Recent advances in electrocatalytic generation of indole-derived radical cations and their applications in organic synthesis;Chinese Chemical Letters;2024-04

2. Integrase;Metalloenzymes;2024

3. The Integrase: An Overview of a Key Player Enzyme in the Antiviral Scenario;International Journal of Molecular Sciences;2023-07-29

4. Base-Controlled Regiospecific Mono-Benzylation/Allylation and Diallylation of 4-Aryl-5-indolyl-1,2,4-triazole-3-thione: Thio-Aza Allyl Rearrangement;Crystals;2023-06-21

5. Synthesis, Characterization and Single Crystal X-ray Diffraction Analysis of Fused Triazolo/Thiadiazole Clubbed with Indole Scaffold;Crystals;2023-03-01