Atom-Economical Synthesis of the N(10)−C(17) Fragment of Cyclotheonamides via a Novel Passerini Reaction−Deprotection−Acyl Migration Strategy1
Author:
Affiliation:
1. Department of Medicinal Chemistry, Corvas International, Inc., 3030 Science Park Road, San Diego, California 92121
Publisher
American Chemical Society (ACS)
Subject
Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry
Link
https://pubs.acs.org/doi/pdf/10.1021/ol0165239
Reference36 articles.
1. Novel, potent and selective chimeric FXa inhibitors featuring hydrophobic p1-ketoamide moieties
2. Synthesis and biological activity of P2–P4 azapeptidomimetic P1-argininal and P1-ketoargininamide derivatives: a novel class of serine protease inhibitors
3. A two-step, one-pot synthesis of diverse N-pyruvoyl amino acid derivatives using the Ugi reaction
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