Microwave-Accelerated Synthesis of P1‘-Extended HIV-1 Protease Inhibitors Encompassing a Tertiary Alcohol in the Transition-State Mimicking Scaffold-Reference-Cited by-同舟云学术

Microwave-Accelerated Synthesis of P1‘-Extended HIV-1 Protease Inhibitors Encompassing a Tertiary Alcohol in the Transition-State Mimicking Scaffold

Published:2006-02-11 Issue:5 Volume:49 Page:1828-1832
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Ekegren Jenny K.¹,Ginman Nina¹,Johansson Åsa¹,Wallberg Hans¹,Larhed Mats¹,Samuelsson Bertil¹,Unge Torsten¹,Hallberg Anders¹

Affiliation:

1. Department of Medicinal Chemistry, Organic Pharmaceutical Chemistry, BMC, Uppsala University, Box 574, SE-751 23 Uppsala, Sweden, Department of Cell and Molecular Biology, Structural Biology, BMC, Uppsala University, Box 596, SE-751 24 Uppsala, Sweden, and Medivir AB, Lunastigen 7, SE-141 44, Huddinge, Sweden

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm051239z

Reference40 articles.

1. Twenty years of therapy for HIV-1 infection

2. New Approaches toward Anti-HIV Chemotherapy

3. Cholinergic activity of acetylenic imidazoles and related compounds

4. HIV-1 protease: mechanism and drug discovery

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