Synthesis and Structure−Activity Relationships of a New Model of Arylpiperazines. 5. Study of the Physicochemical Influence of the Pharmacophore on 5-HT1A/α1-Adrenergic Receptor Affinity: Synthesis of a New Derivative with Mixed 5-HT1A/D2 Antagonist Properties-Reference-Cited by-同舟云学术

Synthesis and Structure−Activity Relationships of a New Model of Arylpiperazines. 5. Study of the Physicochemical Influence of the Pharmacophore on 5-HT1A/α1-Adrenergic Receptor Affinity: Synthesis of a New Derivative with Mixed 5-HT1A/D2 Antagonist Properties

Published:2000-12-21 Issue:2 Volume:44 Page:186-197
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

López-Rodríguez María L.¹,Morcillo M. José¹,Fernández Esther¹,Porras Esther¹,Orensanz Luis¹,Beneytez M Eugenia¹,Manzanares Jorge¹,Fuentes Jose Angel¹

Affiliation:

1. Departamento de Química Orgánica I, Facultad de Ciencias Químicas, and Departamento de Farmacología, Facultad de Farmacia, Universidad Complutense, 28040 Madrid, Spain, Facultad de Ciencias, Universidad Nacional de Educación a Distancia, 28040 Madrid, Spain, and Hospital Ramón y Cajal, Carretera de Colmenar km. 9, 28034 Madrid, Spain

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm000929u

Reference41 articles.

1. 5-HT Receptor Classification and Nomenclature: Towards a Harmonization with the Human Genome

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