Process Development Challenges to Accommodate A Late-Appearing Stable Polymorph: A Case Study on the Polymorphism and Crystallization of a Fast-Track Drug Development Compound-Reference-Cited by-同舟云学术

Process Development Challenges to Accommodate A Late-Appearing Stable Polymorph: A Case Study on the Polymorphism and Crystallization of a Fast-Track Drug Development Compound

Published:2005-11-01 Issue:6 Volume:9 Page:933-942
ISSN:1083-6160
Container-title:Organic Process Research & Development
language:en
Short-container-title:Org. Process Res. Dev.

Author:

Desikan Sridhar¹,Parsons, Rodney L.¹,Davis Wayne P.¹,Ward James E.¹,Marshall Will J.¹,Toma Pascal H.¹

Affiliation:

1. Pharmaceutical Research Institute, Bristol Myers Squibb Company, New Brunswick, New Jersey 08903, U.S.A.

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/op0501287

Reference8 articles.

1. Disappearing Polymorphs

2. Dealing with the Impact of Ritonavir Polymorphs on the Late Stages of Bulk Drug Process Development

3. General Scope of 1,4-Diastereoselective Additions to a 2(3H)-Quinazolinone: Practical Preparation of HIV Therapeutics

4. A new asymmetric 1,4-addition method: application to the synthesis of the HIV non-nucleoside reverse transcriptase inhibitor DPC 961

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