Potent Nonpeptide Antagonists of the Bradykinin B1 Receptor: Structure−Activity Relationship Studies with Novel Diaminochroman Carboxamides-Reference-Cited by-同舟云学术

Potent Nonpeptide Antagonists of the Bradykinin B1 Receptor: Structure−Activity Relationship Studies with Novel Diaminochroman Carboxamides

Published:2007-04-05 Issue:9 Volume:50 Page:2200-2212
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Biswas Kaustav¹,Li Aiwen¹,Chen Jian Jeffrey¹,D'Amico Derin C.¹,Fotsch Christopher¹,Han Nianhe¹,Human Jason¹,Liu Qingyian¹,Norman Mark H.¹,Riahi Bobby¹,Yuan Chester¹,Suzuki Hideo¹,Mareska David A.¹,Zhan James¹,Clarke David E.¹,Toro Andras¹,Groneberg Robert D.¹,Burgess Laurence E.¹,Lester-Zeiner Dianna¹,Biddlecome Gloria¹,Manning Barton H.¹,Arik Leyla¹,Dong Hong¹,Huang Ming¹,Kamassah Augustus¹,Loeloff Richard¹,Sun Hong¹,Hsieh Feng-Yin¹,Kumar Gondi¹,Ng Gordon Y.¹,Hungate Randall W.¹,Askew Benny C.¹,Johnson Eileen¹

Affiliation:

1. Departments of Chemistry Research and Discovery, Pharmacokinetics and Drug Metabolism, Neuroscience, and Inflammation, Amgen Inc., One Amgen Center Drive, Thousand Oaks, California 91320, and Array BioPharma, 3200 Walnut Street, Boulder, Colorado 80301

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm070055c

Reference41 articles.

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5. Kinin receptors

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