General and Scalable Amide Bond Formation with Epimerization-Prone Substrates Using T3P and Pyridine
Author:
Affiliation:
1. Pfizer Worldwide Research and Development, Eastern Point Road, Groton, Connecticut 06340, United States
Publisher
American Chemical Society (ACS)
Subject
Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry
Link
https://pubs.acs.org/doi/pdf/10.1021/ol201875q
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1. A Knowledge-Based Approach in Designing Combinatorial or Medicinal Chemistry Libraries for Drug Discovery. 1. A Qualitative and Quantitative Characterization of Known Drug Databases
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3. Evolution of amide bond formation
4. Amide bond formation: beyond the myth of coupling reagents
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