Covalent Allosteric Inactivation of Protein Tyrosine Phosphatase 1B (PTP1B) by an Inhibitor–Electrophile Conjugate-Reference-Cited by-同舟云学术

Covalent Allosteric Inactivation of Protein Tyrosine Phosphatase 1B (PTP1B) by an Inhibitor–Electrophile Conjugate

Published:2017-04-03 Issue:14 Volume:56 Page:2051-2060
ISSN:0006-2960
Container-title:Biochemistry
language:en
Short-container-title:Biochemistry

Author:

Punthasee Puminan¹,Laciak Adrian R.¹,Cummings Andrea H.¹,Ruddraraju Kasi Viswanatharaju¹,Lewis Sarah M.¹,Hillebrand Roman¹,Singh Harkewal¹,Tanner John J.¹²,Gates Kent S.¹²^ORCID

Affiliation:

1. Department of Chemistry, University of Missouri, 125 Chemistry Building, Columbia, Missouri 65211, United States

2. Department of Biochemistry, University of Missouri, 117 Schweitzer Hall, Columbia, Missouri 65211, United States

Funder

Diabetes Action Foundation

Publisher

American Chemical Society (ACS)

Subject

Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.biochem.7b00151

Reference54 articles.

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4. Structural Bioinformatics-Based Design of Selective, Irreversible Kinase Inhibitors

5. Covalent modification with concomitant inactivation of the cAMP-dependent protein kinase by affinity labels containing only L-amino acids

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