A Covalently Attached Progesterone Molecule Outcompetes the Binding of Free Progesterone at an Allosteric Site of Cytochrome P450 3A4-Reference-Cited by-同舟云学术

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A Covalently Attached Progesterone Molecule Outcompetes the Binding of Free Progesterone at an Allosteric Site of Cytochrome P450 3A4

Published:2019-05-14 Issue:6 Volume:30 Page:1629-1635
ISSN:1043-1802
Container-title:Bioconjugate Chemistry
language:en
Short-container-title:Bioconjugate Chem.

Author:

Ducharme Julie¹,Polic Vanja¹,Auclair Karine¹^ORCID

Affiliation:

1. Department of Chemistry, McGill University, Montreal, Quebec, Canada H3A 0B8

Funder

Natural Sciences and Engineering Research Council of Canada

Center in Green Chemistry and catalysis

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Pharmaceutical Science,Pharmacology,Biomedical Engineering,Bioengineering,Biotechnology

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.bioconjchem.9b00248

Reference31 articles.

1. The Underappreciated Role of Allostery in the Cellular Network

2. The ensemble nature of allostery

3. CYTOCHROME P-450 3A4: Regulation and Role in Drug Metabolism

4. Structural basis for ligand promiscuity in cytochrome P450 3A4

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1. Unraveling the Ligand-Binding Sites of CYP3A4 by Molecular Dynamics Simulations with Solvent Probes;Journal of Chemical Information and Modeling;2024-04-09

2. High-throughput assay to simultaneously evaluate activation of CYP3A and the direct and time-dependent inhibition of CYP3A, CYP2C9, and CYP2D6 using liquid chromatography-tandem mass spectrometry;Xenobiotica;2024-02

3. Impact of Heterotropic Allosteric Modulation on the Time-Dependent Inhibition of Cytochrome P450 3A4;DRUG METAB DISPOS;2023

4. Human cytochrome P450 3A7 binding four copies of its native substrate dehydroepiandrosterone 3-sulfate;Journal of Biological Chemistry;2023-08

5. Impact of Heterotropic Allosteric Modulation on the Time-Dependent Inhibition of Cytochrome P450 3A4;Drug Metabolism and Disposition;2023-07-31

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