Novel Nonimidazole Histamine H3 Receptor Antagonists: 1-(4-(Phenoxymethyl)benzyl)piperidines and Related Compounds-Reference-Cited by-同舟云学术

Novel Nonimidazole Histamine H3 Receptor Antagonists: 1-(4-(Phenoxymethyl)benzyl)piperidines and Related Compounds

Published:2003-03-07 Issue:8 Volume:46 Page:1523-1530
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Mikó Tibor¹,Ligneau Xavier¹,Pertz Heinz H.¹,Ganellin C. Robin¹,Arrang Jean-Michel¹,Schwartz Jean-Charles¹,Schunack Walter¹,Stark Holger¹

Affiliation:

1. Institut für Pharmazie, Freie Universität Berlin, Königin-Luise-Strasse 2+4, 14195 Berlin, Germany, Bioprojet Biotech, 4 rue du Chesnay Beauregard BP 96205, 35762 Saint Grégoire Cedex, France, Department of Chemistry, Christopher Ingold Laboratories, University College London, 20 Gordon Street, London WC1H 0AJ, U.K.; Unité de Neurobiologie et Pharmacologie Moléculaire, Centre Paul Broca de l'INSERM, 2ter rue d'Alésia, 75014 Paris, France, and Institut für Pharmazeutische Chemie, Johann Wolfgang Goethe...

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm021084k

Reference53 articles.

1. Auto-inhibition of brain histamine release mediated by a novel class (H3) of histamine receptor

2. Autoinhibition of histamine synthesis mediated by presynaptic H3-receptors

3. Autoregulation of histamine release in brain by presynaptic H3-receptors

4. Histamine inhibits dopamine release in the mouse striatum via presynaptic H3 receptors

5. Histamine H3 receptor-mediated inhibition of serotonin release in the rat brain cortex

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