Structure-Based Design, Synthesis, and Evaluation of Peptide-Mimetic SARS 3CL Protease Inhibitors

Author:

Akaji Kenichi12,Konno Hiroyuki3,Mitsui Hironori2,Teruya Kenta2,Shimamoto Yasuhiro2,Hattori Yasunao2,Ozaki Takeshi4,Kusunoki Masami5,Sanjoh Akira6

Affiliation:

1. Department of Medicinal Chemistry, Kyoto Pharmaceutical University, Yamashina-ku, Kyoto 607-8412, Japan

2. Department of Chemistry, Graduate School of Medical Science, Kyoto Prefectural University of Medicine, Kita-ku, Kyoto 603-8334, Japan

3. Yamagata University, Yonezawa, Yamagata 992-8510, Japan

4. Institute for Protein Research, Osaka University, Suita, Osaka 565-0871, Japan

5. University of Yamanashi, Kofu, Yamanashi 400-8511, Japan

6. R&D Center, Protein Wave Co., Nara 631-0006, Japan

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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