Structure-Based Design and Biological Evaluation of Novel Caspase-2 Inhibitors Based on the Peptide AcVDVAD-CHO and the Caspase-2-Mediated Tau Cleavage Sequence YKPVD314

Author:

Bresinsky Merlin1,Strasser Jessica M.2,Vallaster Bernadette1,Liu Peng3ORCID,McCue William M.4,Fuller Jessica2ORCID,Hubmann Alexander1,Singh Gurpreet2ORCID,Nelson Kathryn M.2ORCID,Cuellar Matthew E.2ORCID,Wilmot Carrie M.5ORCID,Finzel Barry C.4ORCID,Ashe Karen H.3,Walters Michael A.2ORCID,Pockes Steffen123ORCID

Affiliation:

1. Institute of Pharmacy, University of Regensburg, Universitätsstraße 31, Regensburg 93053, Germany

2. Department of Medicinal Chemistry, Institute for Therapeutics Discovery and Development, University of Minnesota, Minneapolis, Minnesota 55414, United States

3. Department of Neurology, University of Minnesota, 2101 6th Street SE, Minneapolis 55455, United States

4. Department of Medicinal Chemistry, University of Minnesota, Minneapolis, Minnesota 55414, United States

5. Department of Biochemistry, Molecular Biology and Biophysics, University of Minnesota, Minneapolis, Minnesota 55455, United States

Funder

National Institute on Aging

Lucas Brothers Foundation

Publisher

American Chemical Society (ACS)

Subject

Pharmacology (medical),Pharmacology

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