Preparation, Biological Evaluation, and First-in-Human Single-Photon Emission Computed Tomography (SPECT) Study of 99mTc-Labeled Prostate-Specific Membrane Antigen (PSMA)-Targeted Radiotracers Containing Triazole with Reduced Kidneys Accumulation

Author:

Xiao Di1,Han Peiwen1,Jiang Yuhao1,Duan Xiaojiang2,Ruan Qing1,Zhang Zhanbin1,Chen Xiaoliang34,Zhang Junbo1ORCID

Affiliation:

1. Key Laboratory of Radiopharmaceuticals of the Ministry of Education, NMPA Key Laboratory for Research and Evaluation of Radiopharmaceuticals (National Medical Products Administration), College of Chemistry, Beijing Normal University, Beijing 100875, P.R. China

2. Department of Nuclear Medicine, Peking University First Hospital, Beijing 100034, P.R. China

3. Department of Nuclear Medicine, Chongqing University Cancer Hospital, Chongqing 400030, P.R. China

4. Hubei Province Key Laboratory of Molecular Imaging, Union Hospital, Tongji Medical College, Huazhong University of Science and Technology, Wuhan 430022, P.R. China

Funder

Beijing Municipal Natural Science Foundation

National Natural Science Foundation of China

Beijing Nova Program

Publisher

American Chemical Society (ACS)

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