Translational Preclinical PET Imaging and Metabolic Evaluation of a New Cannabinoid 2 Receptor (CB2R) Radioligand, (Z)-N-(3-(2-(2-[18F]Fluoroethoxy)ethyl)-4,5-dimethylthiazol-2(3H)-ylidene)-2,2,3,3-tetramethylcyclopropane-1-carboxamide-Reference-Cited by-同舟云学术

Translational Preclinical PET Imaging and Metabolic Evaluation of a New Cannabinoid 2 Receptor (CB₂R) Radioligand, (Z)-N-(3-(2-(2-[¹⁸F]Fluoroethoxy)ethyl)-4,5-dimethylthiazol-2(3H)-ylidene)-2,2,3,3-tetramethylcyclopropane-1-carboxamide

Published:2024-09-13 Issue: Volume: Page:
ISSN:2575-9108
Container-title:ACS Pharmacology & Translational Science
language:en
Short-container-title:ACS Pharmacol. Transl. Sci.

Author:

Auvity Sylvain¹²³,Attili Bala⁴,Caillé Fabien¹^ORCID,Goislard Maud¹,Cayla Jérôme¹,Hinnen Françoise¹,Demphel Stéphane¹,Brulon Vincent¹,Bottlaender Michel¹⁵,Leroy Claire¹,Bormans Guy⁴^ORCID,Kuhnast Bertrand¹^ORCID,Peyronneau Marie-Anne¹^ORCID

Affiliation:

1. CEA, INSERM, CNRS, BioMaps, Service Hospitalier Frédéric Joliot, Université Paris-Saclay, 91400 Orsay, France

2. Inserm UMR-S 1144, Faculté de Pharmacie de Paris, Université Paris-Cité, 75006 Paris, France

3. Assistance Publique-Hôpitaux de Paris, Hôpital Universitaire Necker-Enfants Malades, 75015 Paris, France

4. Laboratory for Radiopharmaceutical Research, Department of Pharmaceutical and Pharmacological Sciences, KU Leuven, 3000 Leuven, Belgium

5. UNIACT, Neurospin, CEA, 91191 Gif-sur-Yvette, France

Publisher

American Chemical Society (ACS)

Link

https://pubs.acs.org/doi/pdf/10.1021/acsptsci.4c00348

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5. Cannabinoid CB2 receptors in human brain inflammation