Series of (([1,1′-Biphenyl]-2-yl)methyl)sulfinylalkyl Alicyclic Amines as Novel and High Affinity Atypical Dopamine Transporter Inhibitors with Reduced hERG Activity-Reference-Cited by-同舟云学术

Series of (([1,1′-Biphenyl]-2-yl)methyl)sulfinylalkyl Alicyclic Amines as Novel and High Affinity Atypical Dopamine Transporter Inhibitors with Reduced hERG Activity

Published:2024-01-05 Issue: Volume: Page:
ISSN:2575-9108
Container-title:ACS Pharmacology & Translational Science
language:en
Short-container-title:ACS Pharmacol. Transl. Sci.

Author:

Ku Therese C.¹^ORCID,Cao Jianjing¹,Won Sung Joon¹,Guo Jiqing²,Camacho-Hernandez Gisela A.¹,Okorom Amarachi V.¹,Salomon Kristine Walloe³^ORCID,Lee Kuo Hao¹,Loland Claus J.³^ORCID,Duff Henry J.³,Shi Lei¹^ORCID,Newman Amy Hauck¹^ORCID

Affiliation:

1. Molecular Targets and Medications Discovery Branch, National Institute on Drug Abuse–Intramural Research Program, National Institutes of Health, 333 Cassell Drive, Baltimore, Maryland 21224, United States

2. Faculty of Medicine, Libin Institute, Calgary T2N 4N1, Canada

3. Laboratory for Membrane Protein Dynamics, Department of Neuroscience, Faculty of Health and Medical Sciences, University of Copenhagen, Blegdamsvej 3, DK-2200 Copenhagen, Denmark

Funder

Natur og Univers, Det Frie Forskningsr?d

National Institute on Drug Abuse

Lundbeck Foundation

Publisher

American Chemical Society (ACS)

Subject

Pharmacology (medical),Pharmacology

Link

https://pubs.acs.org/doi/pdf/10.1021/acsptsci.3c00322

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