Design and Synthesis of Quinoxaline Hybrids as Modulators of HIF-1a, VEGF, and p21 for Halting Colorectal Cancer

Author:

Ayoup Mohammed Salah12ORCID,Rabee Ahmed R.2,Abdel-Hamid Hamida2,Amer Adel2,Abu-Serie Marwa M.3,Ashraf Samah4,Ghareeb Doaa A.45ORCID,Ibrahim Rabab S.6,Hawsawi Mohammed B.7ORCID,Negm Amr18ORCID,Ismail Magda M. F.6

Affiliation:

1. Department of Chemistry, College of Science, King Faisal University, Al-Ahsa 31982, Saudi Arabia

2. Chemistry Department, Faculty of Science, Alexandria University, P.O. Box 426, Alexandria 21321, Egypt

3. Medical Biotechnology Department, Genetic Engineering and Biotechnology Research Institute, City of Scientific Research and Technological Applications (SRTA-City), New Borg El Arab, Alexandria 21934, Egypt

4. Bio-screening and Preclinical Trial Lab, Biochemistry Department, Faculty of Science, Alexandria University, 21511 Alexandria, Egypt

5. Center of Excellence for Drug Preclinical Studies (CE-DPS), Pharmaceutical and Fermentation Industry Development Center, City of Scientific Research & Technological Applications (SRTA-city), New Borg El Arab, Alexandria 21934, Egypt

6. Department of Pharmaceutical Medicinal Chemistry and Drug Design, Faculty of Pharmacy (Girls), Al-Azhar University, Cairo 11754, Egypt

7. Department of Chemistry, Faculty of Science, Umm Al-Qura University, Al Taif Road, Makkah 24382, Saudi Arabia

8. Chemistry Department, Faculty of Science, Mansoura University, Mansoura 35516, Egypt

Funder

Deanship of Scientific Research, King Faisal University

Publisher

American Chemical Society (ACS)

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