Inhibition of the RNA-Dependent RNA-Polymerase from SARS-CoV-2 by 6-Chloropurine Isoxazoline-Carbocyclic Monophosphate Nucleotides

Author:

Leusciatti Marco1,Macchi Beatrice2,Marino-Merlo Francesca3,Mastino Antonio4,Morra Giulia5,Quadrelli Paolo1ORCID

Affiliation:

1. Department of Chemistry, University of Pavia, Viale Taramelli 12, 27100 Pavia,Italy

2. Department of Chemical Science and Technology, University of Rome Tor Vergata, Via della ricerca scientifica 1, 00133 Roma, Italy

3. Department of Chemical, Biological, Pharmaceutical, and Environmental Sciences, University of Messina, Viale Ferdinando Stagno d’Alcontres, 31, 98166 Messina, Italy

4. The Institute of Translational Pharmacology, CNR, Via Fosso del Cavaliere 100, 00133 Roma, Italy

5. Biocomputing Lab, SCITEC-Istituto di Scienze e Tecnologie Chimiche CNR, Via Mario Bianco 9, 20131 Milano, Italy

Funder

Universit? degli Studi di Pavia

Curia S.r.l.

Steroid S.p.A.

Publisher

American Chemical Society (ACS)

Subject

General Chemical Engineering,General Chemistry

Reference28 articles.

1. Severe acute respiratory syndrome coronavirus 2 (SARS-CoV-2) and coronavirus disease-2019 (COVID-19): The epidemic and the challenges

2. WHO announces COVID-19 outbreak a pandemic. http://www.euro.who.int/en/health-topics/healthemergencies/coronavirus-covid-19/news/news/2020/3/whoannounces-covid-19-outbreak-a-pandemic (accessed Sep 7, 2020)

3. Coronavirus (COVID-19) Events As They Happen; WHO, 2019; https://www.who.int/emergencies/diseases/novel-coronavirus-2019/events-as-they-happen (accessed Sep 28, 2020).

4. a COVID-19 Vaccine Development Pipeline; Vaccine Centre, London School of Hygiene and Tropical Medicine . https://vac-lshtm.shinyapps.io/ncov_vaccine_landscape/ (accessed Sep 7, 2020).

5. b COVID-19 Vaccine Tracker. Lay summary. https://covid-19tracker.milkeninstitute.org/ (accessed Sep 7, 2020).

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