Development of BODIPY FL VH032 as a High-Affinity and Selective von Hippel–Lindau E3 Ligase Fluorescent Probe and Its Application in a Time-Resolved Fluorescence Resonance Energy-Transfer Assay
Author:
Affiliation:
1. Department of Chemical Biology and Therapeutics, St. Jude Children’s Research Hospital, 262 Danny Thomas Place, Mail Stop 1000, Memphis, Tennessee 38105, United States
Publisher
American Chemical Society (ACS)
Subject
General Chemical Engineering,General Chemistry
Link
http://pubs.acs.org/doi/pdf/10.1021/acsomega.0c05221
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1. Binding of the von Hippel-Lindau Tumor Suppressor Protein to Elongin B and C
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3. The tumour suppressor protein VHL targets hypoxia-inducible factors for oxygen-dependent proteolysis
4. Targeting the von Hippel–Lindau E3 Ubiquitin Ligase Using Small Molecules To Disrupt the VHL/HIF-1α Interaction
5. Small-Molecule Inhibitors of the Interaction between the E3 Ligase VHL and HIF1α
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