Rational Design of Novel Anticancer Small-Molecule RNA m6A Demethylase ALKBH5 Inhibitors
Author:
Affiliation:
1. Institute of Chemistry, University of Tartu, Ravila 14a, Tartu 50411, Estonia
2. Chemestmed, Ltd., Riia tn 130b/2, Tartu 50411, Estonia
3. Faculty of Medicine, Department of Pharmacology, University of Helsinki, Helsinki 00014, Finland
Funder
Chemestmed, Ltd.
Publisher
American Chemical Society (ACS)
Subject
General Chemical Engineering,General Chemistry
Link
https://pubs.acs.org/doi/pdf/10.1021/acsomega.1c01289
Reference64 articles.
1. Chemical Modifications to RNA: A New Layer of Gene Expression Regulation
2. Epigenetic Modifications of mRNA and DNA in Plants
3. Dynamic RNA Modifications in Gene Expression Regulation
4. The Dark Side of the Epitranscriptome: Chemical Modifications in Long Non-Coding RNAs
5. Dynamic transcriptomic m6A decoration: writers, erasers, readers and functions in RNA metabolism
Cited by 55 articles. 订阅此论文施引文献 订阅此论文施引文献,注册后可以免费订阅5篇论文的施引文献,订阅后可以查看论文全部施引文献
1. EGFR promotes ALKBH5 nuclear retention to attenuate N6-methyladenosine and protect against ferroptosis in glioblastoma;Molecular Cell;2023-12
2. The role of m6A demethylases in lung cancer: diagnostic and therapeutic implications;Frontiers in Immunology;2023-11-29
3. Discovery of Pyrazolo[1,5-a]pyrimidine Derivative as a Novel and Selective ALKBH5 Inhibitor for the Treatment of AML;Journal of Medicinal Chemistry;2023-11-20
4. Low expression of ZFP36L1 in osteosarcoma promotes lung metastasis by inhibiting the SDC4-TGF-β signaling feedback loop;Oncogene;2023-11-07
5. Dynamic alterations of the transcriptome-wide m6A methylome in cytogenetically normal acute myeloid leukaemia during initial diagnosis and relapse;Genomics;2023-11
1.学者识别学者识别
2.学术分析学术分析
3.人才评估人才评估
"同舟云学术"是以全球学者为主线,采集、加工和组织学术论文而形成的新型学术文献查询和分析系统,可以对全球学者进行文献检索和人才价值评估。用户可以通过关注某些学科领域的顶尖人物而持续追踪该领域的学科进展和研究前沿。经过近期的数据扩容,当前同舟云学术共收录了国内外主流学术期刊6万余种,收集的期刊论文及会议论文总量共计约1.5亿篇,并以每天添加12000余篇中外论文的速度递增。我们也可以为用户提供个性化、定制化的学者数据。欢迎来电咨询!咨询电话:010-8811{复制后删除}0370
www.globalauthorid.com
TOP
Copyright © 2019-2024 北京同舟云网络信息技术有限公司 京公网安备11010802033243号 京ICP备18003416号-3