Discovery of a Novel Class of Dual GPBAR1 Agonists–RORγt Inverse Agonists for the Treatment of IL-17-Mediated Disorders

Author:

Fiorillo Bianca1ORCID,Roselli Rosalinda1,Finamore Claudia1,Biagioli Michele2,di Giorgio Cristina2,Bordoni Martina3,Conflitti Paolo4,Marchianò Silvia2,Bellini Rachele2,Rapacciuolo Pasquale1,Cassiano Chiara1,Limongelli Vittorio14ORCID,Sepe Valentina1ORCID,Catalanotti Bruno1ORCID,Fiorucci Stefano2,Zampella Angela1ORCID

Affiliation:

1. Department of Pharmacy, University of Naples “Federico II”, Via D. Montesano, 49, I-80131 Naples, Italy

2. Department of Medicine and Surgery, University of Perugia, Piazza L. Severi, 1-06132 Perugia, Italy

3. Precision BioTherapeutics, Srl, Perugia 06128, Italy

4. Faculty of Biomedical Sciences, Euler Institute, Università della Svizzera italiana (USI), via G. Buffi 13, CH-6900 Lugano, Switzerland

Funder

Centro Svizzero di Calcolo Scientifico

Universit? degli Studi di Napoli Federico II

H2020 European Research Council

Ministero dell'Istruzione, dell'Universit? e della Ricerca

Publisher

American Chemical Society (ACS)

Subject

General Chemical Engineering,General Chemistry

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