Discovery of a Novel Non-Narcotic Analgesic Derived from the CL-20 Explosive: Synthesis, Pharmacology, and Target Identification of Thiowurtzine, a Potent Inhibitor of the Opioid Receptors and the Ion Channels-Reference-Cited by-同舟云学术

Discovery of a Novel Non-Narcotic Analgesic Derived from the CL-20 Explosive: Synthesis, Pharmacology, and Target Identification of Thiowurtzine, a Potent Inhibitor of the Opioid Receptors and the Ion Channels

Published:2021-05-31 Issue:23 Volume:6 Page:15400-15411
ISSN:2470-1343
Container-title:ACS Omega
language:en
Short-container-title:ACS Omega

Author:

Aguero Stephanie¹,Megy Simon¹,Eremina Valeria V.²,Kalashnikov Alexander I.²,Krylova Svetlana G.³,Kulagina Daria A.²,Lopatina Ksenia A.³,Fournier Mailys¹,Povetyeva Tatyana N.³,Vorozhtsov Alexander B.⁴,Sysolyatin Sergey V.²,Zhdanov Vadim V.³,Terreux Raphael¹^ORCID

Affiliation:

1. Équipe ECMO, Laboratoire de Biologie Tissulaire et d’Ingénierie (LBTI), UMR5305, Université Lyon 1, Lyon 69367, France

2. Institute for Problems of Chemical and Energetic Technologies, Siberian Branch of the Russian Academy of Sciences (IPCET SB RAS), Biysk 659322, Altai Krai, Russia

3. Goldberg Research Institute of Pharmacology and Regenerative Medicine, Tomsk National Research Medical Center of the Russian Academy of Sciences, Tomsk 634028, Russia

4. National Research Tomsk State University, Lenin Avenue, 36, Tomsk 634050, Russia

Publisher

American Chemical Society (ACS)

Subject

General Chemical Engineering,General Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acsomega.1c01786

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