Phosphorylated Morpholine Acetal Human Neurokinin-1 Receptor Antagonists as Water-Soluble Prodrugs-Reference-Cited by-同舟云学术

Phosphorylated Morpholine Acetal Human Neurokinin-1 Receptor Antagonists as Water-Soluble Prodrugs

Published:2000-02-25 Issue:6 Volume:43 Page:1234-1241
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Hale Jeffrey J.¹,Mills Sander G.¹,MacCoss Malcolm¹,Dorn Conrad P.¹,Finke Paul E.¹,Budhu Richard J.¹,Reamer Robert A.¹,Huskey Su-Er W.¹,Luffer-Atlas Debra¹,Dean Brian J.¹,McGowan Erin M.¹,Feeney William P.¹,Chiu Shuet-Hing Lee¹,Cascieri Margaret A.¹,Chicchi Gary G.¹,Kurtz Marc M.¹,Sadowski Sharon¹,Ber Elzbieta¹,Tattersall F. David¹,Rupniak Nadia M. J.¹,Williams Angela R.¹,Rycroft Wayne¹,Hargreaves Richard¹,Metzger Joseph M.¹,MacIntyre D. Euan¹

Affiliation:

1. Merck Research Laboratories, P.O. Box 2000, Rahway, New Jersey 07065, and Merck, Sharp & Dohme, Neuroscience Research Centre, Terlings Park, Eastwick Road, Harlow, Essex CM20 2QR, U.K.

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm990617v

Reference33 articles.

1. Drug Treatment of Chemotherapy-Induced Delayed Emesis

2. The molecular biology of receptors: Techniques and application of receptor research

3. Towards Understanding the Aetiology and Pathophysiology of the Emetic Reflex: Novel Approaches to Antiemetic Drugs

Cited by 96 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Safety assessment of neurokinin-1 receptor antagonist: real-world adverse event analysis from the FAERS database;Frontiers in Pharmacology;2024-07-31

2. Pharmacokinetics of Novel Dopamine Transporter Inhibitor CE-123 and Modafinil with a Focus on Central Nervous System Distribution;International Journal of Molecular Sciences;2023-11-29

3. Fosaprepitant Weekly vs Every 3 Weeks for the Prevention of Concurrent Chemoradiotherapy–Induced Nausea and Vomiting;JAMA Network Open;2023-07-27

4. Degradable polyprodrugs: design and therapeutic efficiency;Chemical Society Reviews;2022

5. Emerging nanoformulation strategies for phytocompounds and applications from drug delivery to phototherapy to imaging;Bioactive Materials;2021-12