Tyrphostins. 5. Potent Inhibitors of Platelet-Derived Growth Factor Receptor Tyrosine Kinase: Structure−Activity Relationships in Quinoxalines, Quinolines, and Indole Tyrphostins-Reference-Cited by-同舟云学术

Tyrphostins. 5. Potent Inhibitors of Platelet-Derived Growth Factor Receptor Tyrosine Kinase: Structure−Activity Relationships in Quinoxalines, Quinolines, and Indole Tyrphostins

Published:1996-01-01 Issue:11 Volume:39 Page:2170-2177
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Gazit Aviv¹,App Harald¹,McMahon Gerald¹,Chen Jefferey¹,Levitzki Alexander¹,Bohmer Frank D.¹

Affiliation:

1. Department of Biological Chemistry, The Alexander Silverman Institute of Life Sciences, The Hebrew University of Jerusalem, Givat Ram, Jerusalem 91904, Israel, SUGEN, Inc., 515 Galveston Drive, Redwood City, California 94063-4720, and Max-Planck Society, Research Group “Growth Factor Signal Transduction” Medical Faculty, Friedrich-Schiller University, Drackendorfer Str. I D 07747, Germany

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm950727b

Reference31 articles.

1. Platelet-derived growth factor receptor signals.

2. Mice deficient for PDGF B show renal, cardiovascular, and hematological abnormalities.

3. Abnormal kidney development and hematological disorders in PDGF beta-receptor mutant mice.

4. The biology of platelet-derived growth factor

5. Platelet-derived growth factor: mechanism of action and possible in vivo function.

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