A Fluoro Analogue of the Menadione Derivative 6-[2‘-(3‘-Methyl)-1‘,4‘-naphthoquinolyl]hexanoic Acid Is a Suicide Substrate of Glutathione Reductase. Crystal Structure of the Alkylated Human Enzyme-Reference-Cited by-同舟云学术

A Fluoro Analogue of the Menadione Derivative 6-[2‘-(3‘-Methyl)-1‘,4‘-naphthoquinolyl]hexanoic Acid Is a Suicide Substrate of Glutathione Reductase. Crystal Structure of the Alkylated Human Enzyme

Published:2006-07-28 Issue:33 Volume:128 Page:10784-10794
ISSN:0002-7863
Container-title:Journal of the American Chemical Society
language:en
Short-container-title:J. Am. Chem. Soc.

Author:

Bauer Holger¹,Fritz-Wolf Karin¹,Winzer Andreas¹,Kühner Sebastian¹,Little Susan¹,Yardley Vanessa¹,Vezin Hervé¹,Palfey Bruce¹,Schirmer R. Heiner¹,Davioud-Charvet Elisabeth¹

Affiliation:

1. Contribution from the Biochemie-Zentrum der Universität Heidelberg, Im Neuenheimer Feld 504, D-69120 Heidelberg, Germany, Centre National de la Recherche Scientifique, 3 rue Michel-Ange, 75794 Paris cedex 16, France, Max-Planck-Institut für Medizinische Forschung, Jahnstrasse 29, D-69120 Heidelberg, Germany, Department of Infections and Tropical Diseases, London School of Hygiene & Tropical Medicine, Keppel Street, London WC1E 7HT, United Kingdom, Laboratoire de Chimie Organique et Macromoléculaire, UMR...

Publisher

American Chemical Society (ACS)

Subject

Colloid and Surface Chemistry,Biochemistry,General Chemistry,Catalysis

Link

https://pubs.acs.org/doi/pdf/10.1021/ja061155v

Reference52 articles.

1. Kinetic Characterization of Glutathione Reductase from the Malarial Parasite Plasmodium falciparum

2. Disulfide-Reductase Inhibitors as Chemotherapeutic Agents: The Design of Drugs for Trypanosomiasis and Malaria

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