(R)-3,N-Dimethyl-N-[1-methyl-3-(4-methylpiperidin-1-yl)propyl]benzenesulfonamide: The First Selective 5-HT7 Receptor Antagonist-Reference-Cited by-同舟云学术

(R)-3,N-Dimethyl-N-[1-methyl-3-(4-methylpiperidin-1-yl)propyl]benzenesulfonamide: The First Selective 5-HT7 Receptor Antagonist

Published:1998-02-01 Issue:5 Volume:41 Page:655-657
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Forbes Ian T.¹,Dabbs Steven¹,Duckworth D. Malcolm¹,Jennings Andrew J.¹,King Frank D.¹,Lovell Peter J.¹,Brown Anthony M.¹,Collin Lissa¹,Hagan Jim J.¹,Middlemiss Derek N.¹,Riley Graham J.¹,Thomas David R.¹,Upton Neil¹

Affiliation:

1. SmithKline Beecham Pharmaceuticals, New Frontiers Science Park, Third Avenue, Harlow, Essex, England, CM19 5AW

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm970519e

Reference23 articles.

1. A novel adenylyl cyclase-activating serotonin receptor (5-HT7) implicated in the regulation of mammalian circadian rhythms

2. Molecular cloning, characterization, and localization of a high-affinity serotonin receptor (5-HT7) activating cAMP formation.

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