Improved Structure−Activity Relationship Analysis of HIV-1 Protease Inhibitors Using Interaction Kinetic Data
Author:
Affiliation:
1. Department of Biochemistry, Uppsala University, BMC, Box 576, SE-751 23 Uppsala, Sweden, and Medivir AB, Lunastigen 7, SE-141 44 Huddinge, Sweden
Publisher
American Chemical Society (ACS)
Subject
Drug Discovery,Molecular Medicine
Link
https://pubs.acs.org/doi/pdf/10.1021/jm0499110
Reference25 articles.
1. Discovery and optimization of nonpeptide HIV-1 protease inhibitors
2. Stereospecific Synthesis, Structure−Activity Relationship, and Oral Bioavailability of Tetrahydropyrimidin-2-one HIV Protease Inhibitors
3. Design and Fast Synthesis of C-Terminal Duplicated Potent C2-Symmetric P1/P1‘-Modified HIV-1 Protease Inhibitors
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