Potent Macrocyclic Inhibitors of Insulin-Regulated Aminopeptidase (IRAP) by Olefin Ring-Closing Metathesis-Reference-Cited by-同舟云学术

Potent Macrocyclic Inhibitors of Insulin-Regulated Aminopeptidase (IRAP) by Olefin Ring-Closing Metathesis

Published:2011-05-09 Issue:11 Volume:54 Page:3779-3792
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Andersson Hanna¹,Demaegdt Heidi²,Johnsson Anders¹,Vauquelin Georges²,Lindeberg Gunnar¹,Hallberg Mathias³,Erdélyi Máté⁴⁵,Karlén Anders¹,Hallberg Anders¹

Affiliation:

1. Department of Medicinal Chemistry, Uppsala University, Box 574, SE-751 23 Uppsala, Sweden

2. Department of Molecular and Biochemical Pharmacology, Vrije Universiteit Brussel, Pleinlaan 2, 1050 Brussels, Belgium

3. Department of Pharmaceutical Biosciences, Uppsala University, Box 591, SE-751 24 Uppsala, Sweden

4. Department of Chemistry, University of Gothenburg, SE-412 96 Gothenburg, Sweden

5. Swedish NMR Centre, University of Gothenburg, Box 465, SE-405 30 Gothenburg, Sweden

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm200036n

Reference91 articles.

1. Attenuation of scopolamine-induced learning deficits by LVV-hemorphin-7 in rats in the passive avoidance and water maze paradigms

2. Dopamine D4 receptor antagonist L745,870 abolishes cognitive effects of intracerebroventricular angiotensin IV and des-Phe6-Ang IV in rats

3. The 3–7 fragment of angiotensin II is probably responsible for its psychoactive properties

4. Angiotensin ii-(3–8)-hexapeptide affects motor activity, performance of passive avoidance and a conditioned avoidance response in rats

5. Strain differences in the effects of Angiotensin IV on mouse cognition

Cited by 44 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Transition Metal‐Catalyzed Reactions and Solid‐Phase Synthesis: A Convenient Blend;European Journal of Organic Chemistry;2022-08-05

2. Recent Advances in Macrocyclic Drugs and Microwave-Assisted and/or Solid-Supported Synthesis of Macrocycles;Molecules;2022-02-02

3. Microwave-assisted synthesis of medicinally privileged heterocycles;Green Synthetic Approaches for Biologically Relevant Heterocycles;2021

4. From Angiotensin IV to Small Peptidemimetics Inhibiting Insulin-Regulated Aminopeptidase;Frontiers in Pharmacology;2020-10-15

5. IRAP Inhibitors: M1-Aminopeptidase Family Inspiration;Frontiers in Pharmacology;2020-09-25