Fragment-Based Ligand Design of Novel Potent Inhibitors of Tankyrases-Reference-Cited by-同舟云学术

Fragment-Based Ligand Design of Novel Potent Inhibitors of Tankyrases

Published:2013-06-04 Issue:11 Volume:56 Page:4497-4508
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Larsson E. Andreas¹,Jansson Anna¹,Ng Fui Mee²,Then Siew Wen²,Panicker Resmi¹,Liu Boping²,Sangthongpitag Kanda²,Pendharkar Vishal²,Tai Shi Jing²,Hill Jeffrey²,Dan Chen¹,Ho Soo Yei²,Cheong Wei Wen²,Poulsen Anders²,Blanchard Stephanie²,Lin Grace Ruiting²,Alam Jenefer²,Keller Thomas H.²,Nordlund Pär¹³

Affiliation:

1. School of Biological Sciences, Nanyang Technological University, Lab 07-01, 61 Biopolis Drive (Proteos), Singapore 138673

2. Experimental Therapeutics Centre, 31 Biopolis Way, Nanos Level 3, Singapore 138669

3. Department of Medical Biochemistry and Biophysics, Karolinska Institute, Scheeles väg 2, SE-171 77 Stockholm, Sweden

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm400211f

Reference39 articles.

1. Axin2 as regulatory and therapeutic target in newborn brain injury and remyelination

2. Poly(ADP-ribosyl)ation reactions in the regulation of nuclear functions

3. Tankyrase, a Poly(ADP-Ribose) Polymerase at Human Telomeres

4. PARP inhibition: PARP1 and beyond

5. Tankyrase-targeted therapeutics: expanding opportunities in the PARP family

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