Synthesis, Ionotropic Glutamate Receptor Binding Affinity, and Structure−Activity Relationships of a New Set of 4,5-Dihydro-8-heteroaryl-4-oxo-1,2,4-triazolo[1,5-a]quinoxaline-2-carboxylates Analogues of TQX-173-Reference-Cited by-同舟云学术

Synthesis, Ionotropic Glutamate Receptor Binding Affinity, and Structure−Activity Relationships of a New Set of 4,5-Dihydro-8-heteroaryl-4-oxo-1,2,4-triazolo[1,5-a]quinoxaline-2-carboxylates Analogues of TQX-173

Published:2001-08-11 Issue:19 Volume:44 Page:3157-3165
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Catarzi Daniela¹,Colotta Vittoria¹,Varano Flavia¹,Filacchioni Guido¹,Galli Alessandro¹,Costagli Chiara¹,Carlà Vincenzo¹

Affiliation:

1. Dipartimento di Scienze Farmaceutiche, Universita' di Firenze, Via G. Capponi, 9, 50121 Firenze, Italy, and Dipartimento di Farmacologia Preclinica e Clinica, Universita' di Firenze, Viale G. Pieraccini, 6, 50134 Firenze, Italy

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm010862q

Reference28 articles.

1. Ligands for Glutamate Receptors: Design and Therapeutic Prospects

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4. Review Central & Peripheral Nervous Systems: Glycine-site NMDA receptor antagonists

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