Piperazine Derivatives of [1,2,4]Triazolo[1,5-a][1,3,5]triazine as Potent and Selective Adenosine A2a Receptor Antagonists-Reference-Cited by-同舟云学术

Piperazine Derivatives of [1,2,4]Triazolo[1,5-a][1,3,5]triazine as Potent and Selective Adenosine A2a Receptor Antagonists

Published:2004-07-13 Issue:17 Volume:47 Page:4291-4299
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Vu Chi B.¹,Peng Bo¹,Kumaravel Gnanasambandam¹,Smits Glenn¹,Jin Xiaowei¹,Phadke Deepali¹,Engber Thomas¹,Huang Carol¹,Reilly Jennifer¹,Tam Stacy¹,Grant Donna¹,Hetu Gregg¹,Chen Liqing¹,Zhang Jianbo¹,Petter Russell C.¹

Affiliation:

1. Department of Medicinal Chemistry, Biogen Idec, Inc., 14 Cambridge Center, Cambridge, Massachusetts 02142

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm0498405

Reference36 articles.

1. Adenosine receptors and their modulators

2. The discovery and synthesis of highly potent, A 2a receptor agonists

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