Thiazolide Prodrug Esters and Derived Peptides: Synthesis and Activity

Author:

Stachulski Andrew V.1ORCID,Rossignol Jean-Francois2,Pate Sophie1,Taujanskas Joshua1,Iggo Jonathan A.1ORCID,Aerts Rudi3,Pascal Etienne3,Piacentini Sara4,La Frazia Simone4,Santoro M. Gabriella45,van Vooren Lieven6,Sintubin Liesje6,Cooper Mark7,Swift Karl7,O’Neill Paul M.1ORCID

Affiliation:

1. Donnan and Robert Robinson Laboratories, Department of Chemistry, University of Liverpool, Liverpool L69 7ZD, U.K.

2. Romark Laboratories, L.C., Tampa, Florida 33609, United States

3. Romark Belgium BVBA, Roosveld 6, 3400 Landen, Belgium

4. Department of Biology, University of Rome Tor Vergata, 00133 Rome, Italy

5. Institute of Translational Pharmacology, CNR, Area della Ricerca di Roma 2, Via Fosso del Cavaliere, 00133 Roma, Italy

6. Ardena Gent NV, Kleimor 4, 9030 Mariakerke, Belgium

7. Bio-Techne, Avonmouth, Bristol BS11 9QD, U.K.

Funder

Romark Pharmaceuticals

Publisher

American Chemical Society (ACS)

Subject

Pharmaceutical Science,Drug Discovery,Molecular Biology,Biochemistry

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