Preparation and Biological Evaluation of Indole, Benzimidazole, and Thienopyrrole Piperazine Carboxamides: Potent Human Histamine H4 Antagonists-Reference-Cited by-同舟云学术

Preparation and Biological Evaluation of Indole, Benzimidazole, and Thienopyrrole Piperazine Carboxamides: Potent Human Histamine H4 Antagonists

Published:2005-11-23 Issue:26 Volume:48 Page:8289-8298
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Venable Jennifer D.¹,Cai Hui¹,Chai Wenying¹,Dvorak Curt A.¹,Grice Cheryl A.¹,Jablonowski Jill A.¹,Shah Chandra R.¹,Kwok Annette K.¹,Ly Kiev S.¹,Pio Barbara¹,Wei Jianmei¹,Desai Pragnya J.¹,Jiang Wen¹,Nguyen Steven¹,Ling Ping¹,Wilson Sandy J.¹,Dunford Paul J.¹,Thurmond Robin L.¹,Lovenberg Timothy W.¹,Karlsson Lars¹,Carruthers Nicholas I.¹,Edwards James P.¹

Affiliation:

1. Johnson & Johnson Pharmaceutical Research and Development, L.L.C., 3210 Merryfield Row, San Diego, California 92121

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm0502081

Reference35 articles.

1. Histamine H4 and H2 Receptors Control Histamine-Induced Interleukin-16 Release from Human CD8+ T Cells

2. Definition and Antagonism of Histamine H2-receptors

3. Cloning and Functional Expression of the Human Histamine H3Receptor

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