Structure−Activity Relationship Studies Optimizing the Antiproliferative Activity of Novel Cyclic Somatostatin Analogues Containing a Restrained Cyclic β-Amino Acid-Reference-Cited by-同舟云学术

Structure−Activity Relationship Studies Optimizing the Antiproliferative Activity of Novel Cyclic Somatostatin Analogues Containing a Restrained Cyclic β-Amino Acid

Published:2005-03-19 Issue:8 Volume:48 Page:2916-2926
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Sukopp Martin¹,Schwab Richard¹,Marinelli Luciana¹,Biron Eric¹,Heller Markus¹,Várkondi Edit¹,Pap Ákos¹,Novellino Ettore¹,Kéri György¹,Kessler Horst¹

Affiliation:

1. Lehrstuhl für Organische Chemie und Biochemie II, Technische Universität München, Lichtenbergstrasse 4, 85747 Garching, Germany, Cooperative Research Center, Semmelweis University, Rippl-Ronai u. 37, and Peptide Biochemistry Research Group of Hung. Acad. Sci., H-1062 Budapest, Hungary, and Dipartimento di Chimica Farmaceutica e Tossicologica, Università “Federico II” di Napoli, Via Domenico Montesano, 49 Napoli, Italy

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm049500j

Reference47 articles.

1. Hypothalamic Polypeptide That Inhibits the Secretion of Immunoreactive Pituitary Growth Hormone

2. Effects of Somatostatin on Hemostasis in Baboons

3. Inhibition by Somatostatin of Glucagon and Insulin Release from the Perfused Rat Pancreas in Response to Arginine, Isoproterenol and Theophylline: Evidence for a Preferential Effect on Glucagon Secretion

4. Somatostatin and Its Receptor Family

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