Fragment-Based Drug Discovery of 2-Thiazolidinones as Inhibitors of the Histone Reader BRD4 Bromodomain-Reference-Cited by-同舟云学术

Fragment-Based Drug Discovery of 2-Thiazolidinones as Inhibitors of the Histone Reader BRD4 Bromodomain

Published:2013-05-14 Issue:10 Volume:56 Page:3833-3851
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Zhao Lele¹,Cao Danyan¹,Chen Tiantian¹,Wang Yingqing²,Miao Zehong²,Xu Yechun¹,Chen Wuyan¹,Wang Xin¹,Li Yanlian¹,Du Zhiyan¹,Xiong Bing¹,Li Jian³,Xu Chunyan³,Zhang Naixia¹,He Jianhua³,Shen Jingkang¹

Affiliation:

1. Department of Medicinal Chemistry, State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zuchongzhi Road, Shanghai 201203, China

2. Division of Anti-Tumor Pharmacology, State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zuchongzhi Road, Shanghai 201203, China

3. Shanghai Institute of Applied Physics, Chinese Academy of Sciences, 239 Zhangheng Road, Shanghai 201204, China

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm301793a

Reference50 articles.

1. Chromatin Modifications and Their Function

2. Regulation of chromatin by histone modifications

3. Combinatorial complexity in chromatin structure and function: revisiting the histone code

4. Translating the Histone Code

5. The language of covalent histone modifications

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