Binding Thermodynamics as a Tool To Investigate the Mechanisms of Drug−Receptor Interactions: Thermodynamics of Cytoplasmic Steroid/Nuclear Receptors in Comparison with Membrane Receptors-Reference-Cited by-同舟云学术

Binding Thermodynamics as a Tool To Investigate the Mechanisms of Drug−Receptor Interactions: Thermodynamics of Cytoplasmic Steroid/Nuclear Receptors in Comparison with Membrane Receptors

Published:2004-09-21 Issue:6 Volume:48 Page:2026-2035
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Gilli Paola¹,Gilli Gastone¹,Borea Pier Andrea¹,Varani Katia¹,Scatturin Angelo¹,Dalpiaz Alessandro¹

Affiliation:

1. Centro di Strutturistica Diffrattometrica and Dipartimento di Chimica, University of Ferrara, via Borsari 46, 44100, Ferrara, Italy, Dipartimento di Medicina Clinica e Sperimentale, University of Ferrara, via Fossato di Mortara 19, 44100, Ferrara, Italy, Dipartimento di Scienze Farmaceutiche, University of Ferrara, via Fossato di Mortara 19, 44100, Ferrara, Italy, and Interdisciplinary Center for the Study of Inflammation (ICSI), University of Ferrara, via Fossato di Mortara 19, 44100, Ferrara, Italy

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm040842z

Reference87 articles.

1. Raffa, R. B., Ed.Drug-Receptor Thermodynamics: Introduction andApplications; Wiley & Sons: New York, 2001; pp 221−416.

2. Can thermodynamic measurements of receptor binding yield information on drug affinity and efficacy?

3. Do thermodynamic studies provide information on both the binding to and the activation of dopaminergic and other receptors?

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