Total Synthesis of Thiaplakortone A: Derivatives as Metabolically Stable Leads for the Treatment of Malaria-Reference-Cited by-同舟云学术

Total Synthesis of Thiaplakortone A: Derivatives as Metabolically Stable Leads for the Treatment of Malaria

Published:2014-01-02 Issue:2 Volume:5 Page:178-182
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Pouwer Rebecca H.¹,Deydier Sophie M.¹,Le Phuc Van¹,Schwartz Brett D.¹,Franken Nicole C.¹,Davis Rohan A.¹,Coster Mark J.¹,Charman Susan A.²,Edstein Michael D.³,Skinner-Adams Tina S.¹,Andrews Katherine T.¹,Jenkins Ian D.¹,Quinn Ronald J.¹

Affiliation:

1. Eskitis Institute for Drug Discovery, Griffith University, Brisbane, QLD 4111, Australia

2. Centre for Drug Candidate Optimisation, Monash University, 381 Royal Parade, Parkville, VIC 3052, Australia

3. Australian Army Malaria Institute, Brisbane, QLD 4051, Australia

Funder

National Health and Medical Research Council

Australian Research Council

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/ml400447v

Reference32 articles.

1. World Health Organization. World Malaria Report 2011, Geneva. http://www.who.int/malaria/world_malaria_report_2011/WMR2011_noprofiles_lowres.pdf(accessed 27 August 2013) .

2. Changes in the Treatment Responses to Artesunate-Mefloquine on the Northwestern Border of Thailand during 13 Years of Continuous Deployment

3. Artemisinin Resistance inPlasmodium falciparumMalaria

4. Challenges facing drug development for malaria

5. Drug-resistant malaria: Molecular mechanisms and implications for public health

Cited by 26 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Synthesis and Antimalarial Evaluation of Halogenated Analogues of Thiaplakortone A;Marine Drugs;2023-05-22

2. Thiaplakortone B attenuates RANKL‐induced NF‐κB and MAPK signaling and dampens OVX‐induced bone loss in mice;Biomedicine & Pharmacotherapy;2022-10

3. Australian chemistry and drug discovery towards the development of antimalarials;Australian Journal of Chemistry;2022-09-02

4. Synthesis, In Silico Studies, and Larvicidal Activity of Novel Hydrazinyl 1,3-Thiazine Derivatives;Russian Journal of Organic Chemistry;2022-06

5. Marine Pyrrole Alkaloids;Marine Drugs;2021-09-10