Unique and Efficient Synthesis of [2S-(2R*,3S*,4R*)]-2-Amino-1-cyclohexyl- 6-methyl-3,4-heptanediol, a Popular C-Terminal Component of Many Renin Inhibitors-Reference-Cited by-同舟云学术

Unique and Efficient Synthesis of [2S-(2R*,3S*,4R*)]-2-Amino-1-cyclohexyl- 6-methyl-3,4-heptanediol, a Popular C-Terminal Component of Many Renin Inhibitors

Published:1996-01-01 Issue:26 Volume:61 Page:9564-9568
ISSN:0022-3263
Container-title:The Journal of Organic Chemistry
language:en
Short-container-title:J. Org. Chem.

Author:

Schwindt Mark A.¹,Belmont Daniel T.¹,Carlson Mark¹,Franklin Lloyd C.¹,Hendrickson Valerie S.¹,Karrick Gregory L.¹,Poe Russell W.¹,Sobieray Denis M.¹,Van De Vusse Jim¹

Affiliation:

1. Chemical Development Department, Parke-Davis Pharmaceutical Research Division, 188 Howard Avenue, Holland, Michigan 49424

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/jo960694n

Reference23 articles.

1. Studies directed toward the design of orally active renin inhibitors. 1. Some factors influencing the absorption of small peptides

2. Stereoselective synthesis of the hydroxy amino acid moiety of Al-77-B, a gastroprotective substance from Bacillus pumilus Al-77

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