A New Efficient Synthetic Route for the Synthesis of the Antiallergic Drug, Olopatadine Hydrochloride, via Stereospecific Palladium-Catalyzed Reaction-Reference-Cited by-同舟云学术

A New Efficient Synthetic Route for the Synthesis of the Antiallergic Drug, Olopatadine Hydrochloride, via Stereospecific Palladium-Catalyzed Reaction

Published:2012-01-12 Issue:2 Volume:16 Page:225-231
ISSN:1083-6160
Container-title:Organic Process Research & Development
language:en
Short-container-title:Org. Process Res. Dev.

Author:

Nishimura Koichiro¹,Kinugawa Masahiko¹

Affiliation:

1. Chemical Process Research and Development Laboratories, Kyowa Hakko Kirin Co., Ltd., 1-1-53, Takasu-cho, Sakai, Osaka 590-8554, Japan

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/op200312m

Reference11 articles.

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3. Katsura, T.; Hayashi, T.; Komatsu, K.; Tanaka, M.PCT Int. Appl. WO/2009/044838 A1, 2009.

4. Bosch, C. J.; Bachs, R. J.; Gomez, G. A.; Alonso, M. Y.; Bessa, S. M.PCT Int. Appl. WO/2006/010459 A1, 2006.

5. Palladium catalysed tandem cyclisation-anion capture processes.Hydride ion capture by vinylpalladium species.

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