2-Carboxyquinoxalines Kill Mycobacterium tuberculosis through Noncovalent Inhibition of DprE1

Author:

Neres João12,Hartkoorn Ruben C.12,Chiarelli Laurent R.13,Gadupudi Ramakrishna45,Pasca Maria Rosalia13,Mori Giorgia13,Venturelli Alberto4,Savina Svetlana16,Makarov Vadim16,Kolly Gaelle S.12,Molteni Elisabetta13,Binda Claudia13,Dhar Neeraj12,Ferrari Stefania45,Brodin Priscille17,Delorme Vincent17,Landry Valérie7,de Jesus Lopes Ribeiro Ana Luisa3,Farina Davide5,Saxena Puneet5,Pojer Florence12,Carta Antonio8,Luciani Rosaria5,Porta Alessio9,Zanoni Giuseppe9,De Rossi Edda13,Costi Maria Paola145,Riccardi Giovanna13,Cole Stewart T.12

Affiliation:

1. More Medicines for Tuberculosis (MM4TB) Consortium ()

2. Global Health Institute, Ecole Polytechnique Fédérale de Lausanne, 1015 Lausanne, Switzerland

3. Department of Biology and Biotecnology “Lazzaro Spallanzani”, University of Pavia, 27100 Pavia, Italy

4. Tydock Pharma, srl Via Campi 183, 41125 Modena, Italy

5. Department of Life Sciences, University of Modena and Reggio Emilia, Via Campi 183, 41126 Modena, Italy

6. A. N. Bakh Institute of Biochemistry, Russian Academy of Science, 119071 Moscow, Russia

7. Inserm U1019 − CNRS UMR 8204, Institut Pasteur de Lille, Université de Lille, 1 rue du Professeur Calmette, 59019, Lille, France

8. Department of Chemistry and Pharmacy, University of Sassari, 07100 Sassari, Italy

9. Department of Chemistry, University of Pavia, 27100 Pavia, Italy

Funder

European Regional Development Fund

European Research Council

Région Nord Pas de Calais

Agence Nationale de la Recherche

European Commission

Publisher

American Chemical Society (ACS)

Subject

Molecular Medicine,General Medicine,Biochemistry

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